Elinogrel

Name: Elinogrel
Brand: Tocris Bioscience
SKU: 5316

Tocris Bioscience, part of Bio-Techne | Catalog # 5316

Citations (4)

COA / SDS

P2Y12 antagonist

Key Product Details

Description:	P2Y₁₂ antagonist
Chemical Name:	5-Chloro-N-[[[4-[6-Fluoro-1,4-dihydro-7-(methylamino)-2,4-dioxo-3(2H)-quinazolinyl]phenyl]amino]carbonyl]-2-thiophenesulfonamide
Purity:	≥97% (HPLC)
Molecular Weight:	523.95

View Full Technical Details for Elinogrel

Technical Data
Citations

Biological Activity for Elinogrel

Elinogrel is a P2Y₁₂ antagonist; exhibits antiplatelet activity.

Compound Libraries for Elinogrel

Elinogrel is also offered as part of the Tocriscreen 2.0 Max. Find out more about compound libraries available from Tocris.

Technical Data for Elinogrel

M. Wt	523.95
Formula	C₂₀H₁₅ClFN₅O₅S₂
Storage	Store at -20°C
Purity	≥97% (HPLC)
CAS Number	936500-94-6
PubChem ID	16066663
InChi Key	LGSDFTPAICUONK-UHFFFAOYSA-N
Smiles	O=C(NS(C4=CC=C(Cl)S4)(=O)=O)NC(C=C3)=CC=C3N2C(C1=CC(F)=C(NC)C=C1NC2=O)=O

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

Solubility for Elinogrel

	Solvent	Max Conc. mg/mL	Max Conc. mM
Solubility
Solubility	DMSO	52.4	100

Preparing Stock Solutions for Elinogrel

The following data is based on the product molecular weight 523.95.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.91 mL	9.54 mL	19.09 mL
5 mM	0.38 mL	1.91 mL	3.82 mL
10 mM	0.19 mL	0.95 mL	1.91 mL
50 mM	0.04 mL	0.19 mL	0.38 mL

Molarity Calculator

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Reconstitution Calculator

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References for Elinogrel

References are publications that support the biological activity of the product.

Cattaneo State of the art of new P2Y12 antagonists. Intern.Emerg.Med. 2010 PMID: 20177818