MRS 2957 triethylammonium salt

Name: MRS 2957 triethylammonium salt
Brand: Tocris Bioscience
SKU: 4260

Tocris Bioscience, part of Bio-Techne | Catalog # 4260

COA / SDS

Potent and selective P2Y6 agonist

Discontinued Product

4260 has been discontinued. View all P2Y Receptor Agonists products.

Key Product Details

Description:	Potent and selective P2Y₆ agonist
Chemical Name:	P¹-[5'(N⁴-Methoxycytidyl)]-P³-(5'-uridyl)-triphosphate tri(triethylammonium) salt
Purity:	≥99% (HPLC)
Molecular Weight:	1042.94

View Full Technical Details for MRS 2957 triethylammonium salt

Technical Data
Citations

Biological Activity for MRS 2957 triethylammonium salt

MRS 2957 triethylammonium salt is a potent P2Y₆ agonist (EC₅₀ = 12 nM). Displays 14- and 66-fold selectivity against P2Y₂ and P2Y₄ receptors respectively.

Technical Data for MRS 2957 triethylammonium salt

M. Wt	1042.94
Formula	C₁₉H₂₈N₅O₂₀P₃.3(C₂H₅)₃N
Storage	Store at -20°C
Purity	≥99% (HPLC)
PubChem ID	90488923
InChi Key	UCQYWKBGVXRIQK-BJFMRLMLSA-N
Smiles	O[C@@H]1[C@@H](N2C(NC(C=C2)=O)=O)O[C@@H](COP(OP(OP(OC[C@H]3O[C@@H](N4C(NC(C=C4)=NOC)=O)[C@H](O)[C@@H]3O)([O-])=O)([O-])=O)([O-])=O)[C@@H]1O.CC[NH+](CC)CC.CC[NH+](CC)CC.CC[NH+](CC)CC

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

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References for MRS 2957 triethylammonium salt

References are publications that support the biological activity of the product.

Maruoka Pyrimidine ribonucleotides with enhanced selectivity as P2Y₆ receptor agonists: novel 4-alkyloxyimino, (S)-methanocarba, and 5'-triphosphate γ-ester modifications. J.Med.Chem. 2010 PMID: 20446735

MRS 2957 triethylammonium salt

Tocris Bioscience, part of Bio-Techne | Catalog # 4260

Key Product Details

Biological Activity for MRS 2957 triethylammonium salt

Technical Data for MRS 2957 triethylammonium salt

Molarity Calculator

Dilution Calculator

Reconstitution Calculator

References for MRS 2957 triethylammonium salt

Product Documents for MRS 2957 triethylammonium salt

COA

Certificate of Analysis

SDS

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