AR-M 1000390 hydrochloride

Name: AR-M 1000390 hydrochloride
Brand: Tocris Bioscience
SKU: 4335

Tocris Bioscience, part of Bio-Techne | Catalog # 4335

Citations (3)

COA / SDS

Low-internalizing δ agonist

Discontinued Product

4335 has been discontinued. View all delta Opioid Receptor Agonists products.

Key Product Details

Description:	Low-internalizing δ agonist
Chemical Name:	N,N-Diethyl-4-(phenyl-4-piperidinylidenemethyl)-benzamide hydrochloride
Purity:	≥97% (HPLC)
Molecular Weight:	384.94

View Full Technical Details for AR-M 1000390 hydrochloride

Technical Data
Citations

Biological Activity for AR-M 1000390 hydrochloride

AR-M 1000390 hydrochloride is a non-peptidic, low-internalizing δ-selective opioid receptor agonist; derivative of SNC 80 (Cat. No. 0764). Does not trigger acute desensitization of the analgesic response; reduces CFA-induced hyperalgesia. Brain penetrant following systemic administration.

Technical Data for AR-M 1000390 hydrochloride

M. Wt	384.94
Formula	C₂₃H₂₈N₂O.HCl
Storage	Store at -20°C
Purity	≥97% (HPLC)
CAS Number	209808-47-9
PubChem ID	76848958
InChi Key	OTXTZCLQEGSAMW-UHFFFAOYSA-N
Smiles	O=C(N(CC)CC)C1=CC=C(/C(C3=CC=CC=C3)=C2\CCNCC2)C=C1.Cl

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

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References for AR-M 1000390 hydrochloride

References are publications that support the biological activity of the product.

Pradhan Ligand-directed trafficking of the δ-opioid receptor in vivo: Two paths toward analgesic tolerance. J.Neurosci. 2010 PMID: 21147985
Marie Pharmacological characterization of AR-M1000390 at human opioid delta receptors. Life Sci. 2003 PMID: 12875901

AR-M 1000390 hydrochloride

Tocris Bioscience, part of Bio-Techne | Catalog # 4335

Key Product Details

Biological Activity for AR-M 1000390 hydrochloride

Technical Data for AR-M 1000390 hydrochloride

Molarity Calculator

Dilution Calculator

Reconstitution Calculator

References for AR-M 1000390 hydrochloride

Product Documents for AR-M 1000390 hydrochloride

COA

Certificate of Analysis

SDS

CONTACT INFORMATION

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