CST 530, Phenol

Name: CST 530, Phenol
Brand: Tocris Bioscience
SKU: 8066

Tocris Bioscience, part of Bio-Techne | Catalog # 8066

COA / SDS

Functionalized IAP ligand for PROTACs®

Key Product Details

Description:	Functionalized IAP ligand for PROTACs^®
Chemical Name:	tert-Butyl ((S)-1-(((S)-1-cyclohexyl-2-((2S,4S)-4-(3-hydroxyphenoxy)-2-(((R)-1,2,3,4-tetrahydronaphthalen-1-yl)carbamoyl)pyrrolidin-1-yl)-2-oxoethyl)amino)-1-oxopropan-2-yl)(methyl)carbamate
Purity:	≥95% (HPLC)
Molecular Weight:	676.86

View Full Technical Details for CST 530, Phenol

Technical Data
Citations

Biological Activity for CST 530, Phenol

CST 530, Phenol is a functionalized IAP (XIAP and cIAP) ligand for PROTAC^® research and development. Supplied with a phenol functional handle for ready conjugation to a linker/target protein ligand. Part of a range of functionalized tool molecules for PROTAC R&D.

Please contact us for SD files of our available Degrader Building Blocks.

PROTAC^® is a registered trademark of Arvinas Operations, Inc., and is used under license.

Usage Guidelines

This product is provided for use in onward chemistry. Suitable solvents can be used.

Technical Data for CST 530, Phenol

M. Wt	676.86
Formula	C₃₈H₅₂N₄O₇
Storage	Store at -20°C
Purity	≥95% (HPLC)
CAS Number	2241489-43-8
PubChem ID	138911358
InChi Key	ZAGJVXJUYODMFQ-QEXUPYAZSA-N
Smiles	CC(C)(C)OC(N(C)[C@@H](C)C(N[C@@H](C1CCCCC1)C(N2[C@@H](C[C@@H](C2)OC3=CC(O)=CC=C3)C(N[C@H]4C5=CC=CC=C5CCC4)=O)=O)=O)=O

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

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References for CST 530, Phenol

References are publications that support the biological activity of the product.

Ng Heterobifunctional ligase recruiters enable pan-degradation of inhibitor of apoptosis proteins. J.Med.Chem. 2023 PMID: 36996313