Kisspeptin 234

Name: Kisspeptin 234
Brand: Tocris Bioscience
SKU: 3881

Tocris Bioscience, part of Bio-Techne | Catalog # 3881

Citations (9)

COA / SDS

Kisspeptin receptor antagonist; kisspeptin 10 (Cat. No. 2570) analog

Key Product Details

Description:	Kisspeptin receptor antagonist; kisspeptin 10 (Cat. No. 2570) analog
Purity:	≥95% (HPLC)
Molecular Weight:	1295.42

View Full Technical Details for Kisspeptin 234

Technical Data
Citations

Biological Activity for Kisspeptin 234

Kisspeptin 234 is a kisspeptin receptor (KISS1, GPR54) antagonist; kisspeptin-10 (Cat. No. 2570) analog. Inhibits kisspeptin-10 stimulation of inositol phosphate (IP) (IC₅₀ = 7 nM) and release of gonadotrophin-releasing hormone (GnRH).

Licensing Information

Sold under license

Technical Data for Kisspeptin 234

M. Wt	1295.42
Formula	C₆₃H₇₈N₁₈O₁₃
Single Letter Sequence	Ac-ANWNGFGWRF-NH2 (Modifications: Ala-1 = D-Ala & N-terminal Ac, Trp-8 = D-Trp, Phe-10 = C-terminal amide)
Storage	Store at -20°C
Purity	≥95% (HPLC)
CAS Number	1145998-81-7
PubChem ID	90488890
InChi Key	IUPKBWSKNCAQJQ-JYYYXURSSA-N
Smiles	C[C@@H](NC(C)=O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CC1=CNC2=C1C=CC=C2)C(=O)N[C@@H](CC(N)=O)C(=O)NCC(=O)N[C@@H](CC1=CC=CC=C1)C(=O)NCC(=O)N[C@H](CC1=CNC2=C1C=CC=C2)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC1=CC=CC=C1)C(N)=O

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

Solubility for Kisspeptin 234

Solubility

Soluble to 1mg/ml in water

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References for Kisspeptin 234

References are publications that support the biological activity of the product.

Roseweir Discovery of potent kisspeptin antagonists delineate physiological mechanisms of gonadototrophin regulation. J.Neurosci. 2009 PMID: 19321788