5-HT2C Receptor Antagonists: Small Molecules and Peptides
5-HT2C is 7TM serotonin receptor that is neuronally expressed in the limbic system of the brain. 5-HT2C is an important pharmacologic target in the treatment of psychosis, schizophrenia, depression, anxiety, and migrane headaches.
5 results for "5-HT2C Receptor Antagonists Small Molecules and Peptides" in Products
5 results for "5-HT2C Receptor Antagonists Small Molecules and Peptides" in Products
5-HT2C Receptor Antagonists: Small Molecules and Peptides
5-HT2C is 7TM serotonin receptor that is neuronally expressed in the limbic system of the brain. 5-HT2C is an important pharmacologic target in the treatment of psychosis, schizophrenia, depression, anxiety, and migrane headaches.
Potent and selective 5-HT2B and 5-HT2C antagonist; orally active
| Chemical Name: | 3,5-Dihydro-5-methyl-N-3-pyridinylbenzo[1,2-b:4,5-b']dipyrrole-1(2H)-carboxamide hydrochloride |
| Purity: | ≥99% (HPLC) |
Dopamine antagonist with some D4 selectivity; also 5-HT2A/2C antagonist
| Chemical Name: | 8-Chloro-11-(4-methyl-1-piperazinyl)-5H-dibenzo[b,e][1,4]diazepine |
| Purity: | ≥99% (HPLC) |
Selective 5-HT2C antagonist; brain penetrant
| Chemical Name: | 6-Chloro-2,3-dihydro-5-methyl-N-[6-[(2-methyl-3-pyridinyl)oxy]-3-pyridinyl]-1H-indole-1-carboxyamide dihydrochloride |
| Purity: | ≥98% (HPLC) |
Selective 5-HT2C antagonist
| Chemical Name: | 8-[5-(2,4-Dimethoxy-5-(4-trifluoromethylphenylsulphonamido)phenyl-5-oxopentyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione hydrochloride |
| Purity: | ≥98% (HPLC) |
5-HT2A and 5-HT2C antagonist; also D2-like partial agonist
| Alternate Names: | CU-32-085 |
| Chemical Name: | N'-[(8-α1,6-dimethylergolin-8-yl]-N,N-dimethylsulfamide hydrochloride |
| Purity: | ≥99% (HPLC) |
