Estrogen and Related Receptor Antagonists: Small Molecules and Peptides
7 results for "Estrogen and Related Receptor Antagonists Small Molecules and Peptides" in Products
7 results for "Estrogen and Related Receptor Antagonists Small Molecules and Peptides" in Products
Estrogen and Related Receptor Antagonists: Small Molecules and Peptides
Estrogen receptor antagonist
Alternate Names: | Fulvestrant |
Chemical Name: | 7α,17β-[9-[(4,4,5,5,5-Pentafluoropentyl)sulfinyl]nonyl]estra-1,3,5(10)-triene-3,17-diol |
Purity: | ≥99% (HPLC) |
Highly selective ERα antagonist
Chemical Name: | 1,3-Bis(4-hydroxyphenyl)-4-methyl-5-[4-(2-piperidinylethoxy)phenol]-1H-pyrazole dihydrochloride |
Purity: | ≥98% (HPLC) |
Selective ERβ antagonist
Chemical Name: | 4-[2-Phenyl-5,7-bis(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-3-yl]phenol |
Purity: | ≥99% (HPLC) |
Potent and selective G protein-coupled estrogen receptor (GPER) antagonist
Chemical Name: | N-[2-Cyclohexyl-4-(1-methylethyl)phenyl]-4-methoxybenzenemethanamine hydrochloride |
Purity: | ≥98% (HPLC) |
High affinity and selective GPER antagonist
Chemical Name: | (3aS*,4R*,9bR*)-4-(6-Bromo-1,3-benzodioxol-5-yl)-3a,4,5,9b-3H-cyclopenta[c]quinoline |
Purity: | ≥99% (HPLC) |
Selective GPER antagonist
Chemical Name: | (±)-(3aR*,4S*,9bS*)-4-(6-Bromo-1,3-benzodioxol-5-yl)-3a,4,5,9b-tetrahydro-8-(1-methylethyl)-3H-cyclopenta[c]quinoline |
Purity: | ≥99% (HPLC) |
ERα antagonist; also activates unfolded protein response; active in vivo
Chemical Name: | 1,3-Dihydro-3,3-bis(4-hydroxyphenyl)-7-methyl-2H-indol-2-one |
Purity: | ≥98% (HPLC) |