NMDA Receptor Antagonists: Small Molecules and Peptides
NMDA receptors (NMDARs) are members of the glutamate-gated ion-channel family and function in synaptic plasticity, neuronal development and excitotoxicity.
34 results for "NMDA Receptor Antagonists Small Molecules and Peptides" in Products
34 results for "NMDA Receptor Antagonists Small Molecules and Peptides" in Products
NMDA Receptor Antagonists: Small Molecules and Peptides
NMDA receptors (NMDARs) are members of the glutamate-gated ion-channel family and function in synaptic plasticity, neuronal development and excitotoxicity.
Potent and selective NMDA receptor antagonist; more active form of DL-AP5
| Alternate Names: | 2-APV,D-APV,D-2-amino-5-phosphonovalerate |
| Chemical Name: | D-(-)-2-Amino-5-phosphonopentanoic acid |
| Purity: | ≥99% (HPLC) |
Non-competitive NMDA antagonist; acts at ion channel site
| Alternate Names: | Dizocilpine |
| Chemical Name: | (5S,10R)-(+)-5-Methyl-10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5,10-imine maleate |
| Purity: | ≥99% (HPLC) |
Non-competitive NMDA receptor antagonist
| Chemical Name: | 2-(2-Chlorophenyl)-2-(methylamino)cyclohexanone hydrochloride |
| Purity: | ≥99% (HPLC) |
Potent and selective NMDA antagonist
| Alternate Names: | DL-APV |
| Chemical Name: | DL-2-Amino-5-phosphonopentanoic acid |
| Purity: | ≥98% (HPLC) |
Potent and selective non-NMDA iGluR antagonist
| Alternate Names: | Cyanquixaline |
| Chemical Name: | 6-Cyano-7-nitroquinoxaline-2,3-dione |
| Purity: | ≥99% (HPLC) |
NMDA antagonist; acts at ion channel site
| Chemical Name: | 3,5-Dimethyl-tricyclo[3.3.1.13,7]decan-1-amine hydrochloride |
Potent and selective NMDA antagonist; sodium salt of DL-AP5
| Chemical Name: | DL-2-Amino-5-phosphonopentanoic acid sodium salt |
| Purity: | ≥98% (HPLC) |
GluN2B-selective NMDA antagonist
| Chemical Name: | (αR,βS)-α-(4-Hydroxyphenyl)-β-methyl-4-(phenylmethyl)-1-piperidinepropanol maleate |
| Purity: | ≥98% (HPLC) |
Potent NMDA antagonist; more active enantiomer of (RS)-CPP
| Chemical Name: | 3-((R)-2-Carboxypiperazin-4-yl)-propyl-1-phosphonic acid |
Potent kynurenine 3-monooxygenase (KMO) inhibitor
| Chemical Name: | 3,4-Dimethoxy-N-[4-(3-nitrophenyl)-2-thiazolyl]benzenesulfonamide |
| Purity: | ≥99% (HPLC) |
Potent NMDA antagonist; acts at glycine site
| Chemical Name: | 5,7-Dichloro-4-hydroxyquinoline-2-carboxylic acid |
| Purity: | ≥98% (HPLC) |
Non-competitive NMDA antagonist; also σ ligand
| Chemical Name: | (1R*,2S*)-erythro-2-(4-Benzylpiperidino)-1-(4-hydroxyphenyl)-1-propanol hemi-(DL)-tartrate |
| Purity: | ≥99% (HPLC) |
GluN1/GluN2A-selective NMDA antagonist
| Chemical Name: | 3-Chloro-4-fluoro-N-[4-[[2-(phenylcarbonyl)hydrazino]carbonyl]benzyl]benzenesulfonamide |
| Purity: | ≥99% (HPLC) |
GluN2B-selective NMDA antagonist
| Alternate Names: | PD 174494,Ro 63-1908 |
| Chemical Name: | 1-[2-(4-Hydroxyphenoxy)ethyl]-4-[(4-methylphenyl)methyl]-4-piperidinol hydrochloride |
| Purity: | ≥99% (HPLC) |
Highly potent NMDA antagonist
| Chemical Name: | trans-2-Carboxy-5,7-dichloro-4-phenylaminocarbonylamino-1,2,3,4-tetrahydroquinoline |
| Purity: | ≥99% (HPLC) |
NMDA antagonist; less active enantiomer of (+)-MK 801
| Chemical Name: | (5R,10S)-(-)-5-Methyl-10,11-dihydro-5H-dibenzo[a,d]cylcohepten-5,10-imine maleate |
| Purity: | ≥99% (HPLC) |
Potent and selective NMDA antagonist; acts at the glycine site
| Alternate Names: | GV 150526A |
| Chemical Name: | 4,6-Dichloro-3-[(1E)-3-oxo-3-(phenylamino)-1-propenyl]-1H-indole-2-carboxylic acid sodium salt |
| Purity: | ≥98% (HPLC) |
Potent NMDA antagonist
| Chemical Name: | (RS)-3-(2-Carboxypiperazin-4-yl)-propyl-1-phosphonic acid |
Potent and selective NMDA antagonist
| Chemical Name: | (E)-(±)-2-Amino-4-methyl-5-phosphono-3-pentenoic acid |
| Purity: | ≥99% (HPLC) |
Potent and selective NMDA antagonist; less active form of DL-AP5
| Chemical Name: | L-(+)-2-Amino-5-phosphonopentanoic acid |
| Purity: | ≥99% (HPLC) |
Potent competitive NMDA antagonist
| Alternate Names: | Midafotel,SDZ EAA 494 |
| Chemical Name: | D-4-[(2E)-3-Phosphono-2-propenyl]-2-piperazinecarboxylic acid |
NMDA antagonist; acts at glycine site
| Chemical Name: | 7-Chloro-4-hydroxy-3-(3-phenoxy)phenyl-2(1H)-quinolinone |
| Purity: | ≥99% (HPLC) |
Potent and selective NMDA antagonist; acts at glycine site
| Alternate Names: | PAMQX |
| Chemical Name: | [(1S)-1-[[(7-Bromo-1,2,3,4-tetrahydro-2,3-dioxo-5-quinoxalinyl)methyl]amino]ethyl]phosphonic acid hydrochloride |
| Purity: | ≥98% (HPLC) |
Potent non-competitive NMDA antagonist; antinociceptive
| Chemical Name: | 2-Amino-2-(2-chlorophenyl)cyclohexanone hydrochloride |
| Purity: | ≥99% (HPLC) |
Potent competitive NMDA antagonist
| Chemical Name: | cis-4-[Phosphomethyl]-piperidine-2-carboxylic acid |
