Other Kinase Inhibitors: Small Molecules and Peptides
43 results for "Other Kinase Inhibitors Small Molecules and Peptides" in Products
43 results for "Other Kinase Inhibitors Small Molecules and Peptides" in Products
Other Kinase Inhibitors: Small Molecules and Peptides
CaM kinase III (eEF-2 kinase) inhibitor
| Chemical Name: | 1-Hexadecyl-2-methyl-3-(phenylmethyl)-1H-imidazolium iodide |
Potent and selective TAK1/MAP3K7 kinase inhibitor
| Chemical Name: | N1-(1-Propyl-1H-benzimidazol-2-yl)-1,3-benzenedicarboxamide |
| Purity: | ≥98% (HPLC) |
Potent and selective TAK1 MAPKKK inhibitor
| Chemical Name: | (3S,5Z,8S,9S,11E)-3,4,9,10-tetrahydro-8,9,16-trihydroxy-14-methoxy-3-methyl-1H-2-benzoxacyclotetradecin-1,7(8H)-dione |
| Purity: | ≥98% (HPLC) |
Potent MSK1 inhibitor; also inhibits other AGC group kinases
| Chemical Name: | 2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-N-4-piperidinyl-1H-imidazo[4,5-c]pyridine-7-methanamine dihydrochloride |
| Purity: | ≥98% (HPLC) |
Serum- and glucocorticoid-regulated kinase (SGK) inhibitor
| Chemical Name: | 2-Cyclopentyl-4-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl-benzoic acid |
| Purity: | ≥97% (HPLC) |
Potent and selective doublecortin like kinase 1/2 (DCLK1/2) inhibitor; orally bioavailable
| Chemical Name: | 5,11-Dihydro-2-[[2-methoxy-4-(4-methyl-1-piperazinyl)phenyl]amino]-11-methyl-5-(2,2,2-trifluoroethyl)-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one |
| Purity: | ≥98% (HPLC) |
Mitochondrial pyruvate dehydrogenase kinase (PDK) inhibitor
| Chemical Name: | Sodium dichloroacetate |
Lysine deficient protein kinase (WNK) signaling inhibitor
| Chemical Name: | 7-Ethoxy-N3-(2-furanylmethyl)-3,9-acridinediamine |
| Purity: | ≥98% (HPLC) |
Potent and selective polynucleotide kinase/phosphatase (PNKP) inhibitor
| Chemical Name: | 4a,7a-Dihydro-2-(1-hydroxyundecyl)-1-[(4-nitrophenyl)amino]-6-phenyl-1H-pyrrolo[3,4-b]pyridine-5,7(2H,6H)-dione |
| Purity: | ≥98% (HPLC) |
Salt inducible kinase (SIK) inhibitor; also ULK1 and 2 inhibitor
| Chemical Name: | N-[3-[[5-Cyclopropyl-2-[[3-(4-morpholinylmethyl)phenyl]amino]-4-pyrimidinyl]amino]propyl]cyclobutanecarboxamide dihydrochloride |
| Purity: | ≥98% (HPLC) |
Potent and selective pyruvate dehydrogenase kinase (PDK) 1/2/3/4 inhibitor
| Chemical Name: | N-[4-(2-Chloro-5-methyl-4-pyrimidinyl)phenyl]-N-[[4-[[(2,2-difluoroacetyl)amino]methyl]phenyl]methyl]-2,4-dihydroxybenzamide |
| Purity: | ≥98% (HPLC) |
TGF-β-activated kinase (TAK1) inhibitor
| Chemical Name: | N-[4-[(4-Ethyl-1-piperazinyl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-(1H-pyrrolo[2,3-b]pyridin-4-yloxy)benzamide |
| Purity: | ≥98% (HPLC) |
Potent and selective PI 4-kinase IIIβ inhibitor
| Chemical Name: | N-[2-[[6-Chloro-3-[3-[(dimethylamino)sulfonyl]phenyl]-2-methylimidazo[1,2-b]pyridazin-8-yl]amino]ethyl]acetamide |
| Purity: | ≥98% (HPLC) |
Ras signaling inhibitor; inhibits Ack1 and GCK
| Chemical Name: | N-[3-[1,4-Dihydro-1-methyl-7-[(6-methyl-3-pyridinyl)amino]-2-oxopyrimido[4,5-d]pyrimidin-3(2H)-yl]-4-methylphenyl]-3-(trifluoromethyl)benzamide |
| Purity: | ≥98% (HPLC) |
Potent and selective MST3 kinase binding inhibitor
| Chemical Name: | 8-(4-Aminobutyl)-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(1,3-dihydroxypropan-2-ylamino)pyrido[2,3-d]pyrimidin-7-one trihydrochloride |
| Purity: | ≥98% (HPLC) |
Multikinase Degrader (PROTAC®)
| Chemical Name: | N-(2-(2-(2-(4-(4-((5-Chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)piperazin-1-yl)ethoxy)ethoxy)ethyl)-2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)amino)acetamide |
| Purity: | ≥98% (HPLC) |
Potent inhibitor of salt-inducible kinases
| Chemical Name: | 3-(2,4-Dimethoxyphenyl)-4-(3-thienyl)-1H-pyrrolo[2,3-b]pyridine |
| Purity: | ≥98% (HPLC) |
PKR inhibitor
| Chemical Name: | 6,8-Dihydro-8-(1H-imidazol-5-ylmethylene)-7H-pyrrolo[2,3-g]benzothiazol-7-one |
| Purity: | ≥98% (HPLC) |
Potent and selective Cdc7 inhibitor
| Alternate Names: | BMS 863233 |
| Chemical Name: | 8-Chloro-2-(2S)-2-pyrrolidinylbenzofuro[3,2-d]pyrimidin-4(3H)-one hydrochloride |
| Purity: | ≥99% (HPLC) |
High affinity cyclin G associated kinase (GAK) inhibitor
| Chemical Name: | 6-Bromo-N-(3,4,5-trimethoxyphenyl)-4-quinolinamine |
| Purity: | ≥99% (HPLC) |
Potent and selective inhibitor of Chk1 and Wee1
| Chemical Name: | 9-Hydroxy-4-phenyl-pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione |
| Purity: | ≥98% (HPLC) |
Potent and selective Lck and Src inhibitor; also inhibits SIK
| Alternate Names: | KIN112 |
| Chemical Name: | 2,6-Dimethylphenyl-N-(2,4-dimethoxyphenyl)-N-[2-[[4-(4-methyl-1-piperazinyl)phenyl]amino]-4-pyrimidinyl]carbamate |
| Purity: | ≥98% (HPLC) |
Potent TAOK inhibitor
| Chemical Name: | N-(2-Oxo-2-((1,2,3,4-tetrahydronaphthalen-1-yl)amino)ethyl)-[1,1'-biphenyl]-4-carboxamide |
| Purity: | ≥98% (HPLC) |
Potent and selective Tpl2 (Cot; MAP3K8) inhibitor
| Chemical Name: | 4-[(3-Chloro-4-fluorophenyl)amino]-6-[(3-pyridinylmethyl)amino]-1,7-naphthyridine-3-carbonitrile |
| Purity: | ≥99% (HPLC) |
Potent and selective MST1/2 inhibitor; orally bioavailable
| Chemical Name: | 4-[(6,10-Dihydro-5,10-dimethyl-6-oxo-5H-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide |
| Purity: | ≥98% (HPLC) |
