Src Family Kinase Inhibitors: Small Molecules and Peptides
20 results for "Src Family Kinase Inhibitors Small Molecules and Peptides" in Products
20 results for "Src Family Kinase Inhibitors Small Molecules and Peptides" in Products
Src Family Kinase Inhibitors: Small Molecules and Peptides
Potent ATP-competitive Src family kinase inhibitor; also AMPK inhibitor; cell permeable
Chemical Name: | 2,3-Dihydro-N,N-dimethyl-2-oxo-3-[(4,5,6,7-tetrahydro-1H-indol-2-yl)methylene]-1H-indole-5-sulfonamide |
Purity: | ≥98% (HPLC) |
Potent, selective Src family kinase inhibitor
Chemical Name: | 3-(4-chlorophenyl) 1-(1,1-dimethylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine |
Purity: | ≥99% (HPLC) |
Potent, selective Src family kinase inhibitor
Chemical Name: | 1-(1,1-Dimethylethyl)-1-(4-methylphenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine |
Purity: | ≥98% (HPLC) |
Src family kinase inhibitor; also inhibits c-Abl
Alternate Names: | 1-NA-PP 1 |
Chemical Name: | 1-(1,1-Dimethylethyl)-3-(1-naphthalenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine |
Purity: | ≥99% (HPLC) |
Inhibitor of Src family kinases
Chemical Name: | 7-[trans-4-(4-Methyl-1-piperazinyl)cyclohexyl]-5-(4-phenoxyphenyl)-7H-Pyrrolo[2,3-d]pyrimidin-4-amine trihydrochloride |
Purity: | ≥98% (HPLC) |
Dual site Src kinase inhibitor
Chemical Name: | 6,7-Dimethoxy-N-(4-phenoxyphenyl)-4-quinazolinamine |
Purity: | ≥99% (HPLC) |
Potent and selective Src tyrosine kinase family inhibitor; anticancer; antiviral; orally bioavailable
Alternate Names: | AZD 0530 |
Chemical Name: | N-(5-Chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methyl-1-piperazinyl)ethoxy]-5-[(tetrahydro-2H-pyran-4-yl)oxy]-4-quinazolinamine |
Purity: | ≥98% (HPLC) |
Potent and selective c-Src inhibitor
Chemical Name: | 1-[3-[1-([1,1'-Biphenyl]-3-ylmethyl)-1H-1,2,3-triazol-5-yl]phenyl]-3-(4-chlorophenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine |
Purity: | ≥98% (HPLC) |
Src tyrosine kinase inhibitor
Chemical Name: | N-(2-Chloro-5-methoxyphenyl)-6-methoxy |
Purity: | ≥99% (HPLC) |
Potent c-SRC kinase inhibitor; also inhibits DDR2, BTK and Syk
Chemical Name: | 3-[[2-[3-(4-Morpholinylmethyl)phenyl]thieno[3,2-b]pyridin-7-yl]amino]phenol dihydrochloride |
Purity: | ≥98% (HPLC) |
Selective and highly potent Fgr and Lyn kinase inhibitor; orally bioavailable
Chemical Name: | 3-[(6,7-Dimethoxy-4-quinazolinyl)oxy]-N-[4-[(4-ethyl-1-piperazinyl)methyl]-3-(trifluoromethyl)phenyl]-4-methylbenzamide dihydrochloride |
Purity: | ≥98% (HPLC) |
Potent Src inhibitor; also inhibits FGFR1, PDGFRβ and Wee1
Chemical Name: | 6-(2,6-Dichlorophenyl)-2-[[4-[2-(diethylamino)ethoxy]phenyl]amino]-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one dihydrochloride |
Purity: | ≥99% (HPLC) |
Highly potent pan-Src/Bcr-Abl inhibitor
Alternate Names: | BMS-354825 |
Chemical Name: | N-(2-Chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyethyl)-1-piperazinyl]-2-methyl-4-pyrimidinyl]amino]-5-thiazolecarboxamide |
Purity: | ≥98% (HPLC) |
UNC119 chaperone-cargo interaction inhibitor; disrupts Src activation
Chemical Name: | Ethyl 4-((3,4-dioxo-2-((2-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)ethyl)amino)cyclobut-1-en-1-yl)amino)piperidine-1-carboxylate hydrochloride |
Purity: | ≥98% (HPLC) |
Dual Src-Abl inhibitor; antiproliferative
Alternate Names: | SKI-606 |
Chemical Name: | 4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methyl-1-piperazinyl)propoxy]-3-quinolinecarbonitrile |
Purity: | ≥99% |
Potent and selective Lck and Src inhibitor; also inhibits SIK
Alternate Names: | KIN112 |
Chemical Name: | 2,6-Dimethylphenyl-N-(2,4-dimethoxyphenyl)-N-[2-[[4-(4-methyl-1-piperazinyl)phenyl]amino]-4-pyrimidinyl]carbamate |
Purity: | ≥98% (HPLC) |
Potent PDGFRα and PDGFRβ inhibitor; also inhibits c-Abl, Lck, c-Src and Fyn kinases
Chemical Name: | N-(3-Fluorophenyl)-1,4-dihydro-6,7-dimethoxyindeno[1,2-c]pyrazol-3-amine |
Purity: | ≥98% (HPLC) |
Potent and selective breast tumor kinase (Brk) inhibitor
Chemical Name: | 3-(9H-Pyrido[2,3-b]indol-4-ylamino)phenol |
Purity: | ≥98% (HPLC) |
Potent Lck inhibitor
Chemical Name: | 6-(2,6-Dimethylphenyl)-2-[[4-(4-methyl-1-pyrimido[5',4':5,6]pyrimido[1,2-a]benzimidazol-5(6H)-one |
Purity: | ≥98% (HPLC) |
Negative control for PP 2 (Cat. No. 1407)
Chemical Name: | 1-Phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine |
Purity: | ≥98% (HPLC) |