DYRK Inhibitors: Small Molecules and Peptides
10 results for "DYRK Inhibitors Small Molecules and Peptides" in Products
10 results for "DYRK Inhibitors Small Molecules and Peptides" in Products
DYRK Inhibitors: Small Molecules and Peptides
Potent and selective DYRK inhibitor; orally bioavailable.
| Chemical Name: | (5Z)-2-[(2,6-Dichlorophenyl)amino]-5-(6-quinoxalinylmethylene)-4(5H)-thiazolone |
| Purity: | ≥95% (HPLC) |
Potent DYRK1B inhibitor
| Chemical Name: | N-[2-Methoxy-4-(4-methyl-1-piperazinyl)phenyl]-4-(1-methyl-1H-pyrrolo[2,3-c]pyridin-3-yl)-2-pyrimidinamine |
| Purity: | ≥98% (HPLC) |
Inhibitor of Clk and DYRK kinases
| Chemical Name: | 5-(1,3-Benzodioxol-5-yl)-N-[(3,5-dichlorophenyl)methyl]-4-pyrimidinamine hydrochloride |
| Purity: | ≥98% (HPLC) |
Potent and selective DYRK1A inhibitor
| Chemical Name: | 7-Methoxy-1-methyl-9H-pyrido[3,4-b]indole |
| Purity: | ≥98% (HPLC) |
DYRK1A/B inhibitor
| Chemical Name: | (1Z)-1-(3-Ethyl-5-hydroxy-2(3H)-benzothiazolylidene)-2-propanone |
| Purity: | ≥98% (HPLC) |
Potent and selective DYRK1A/B inhibitor
| Chemical Name: | N-[2-Chloro-5-[[[(3-chlorophenyl)methyl]amino]carbonyl]phenyl]-7,8-dihydro-2-methoxy-7-oxopyrido[2,3-d]pyrimidine-6-carboxamide |
| Purity: | ≥98% (HPLC) |
Potent and selective pan-CLK inhibitor; also inhibits DYRK1A/B
| Chemical Name: | 4-[1,1-Dimethyl-2-(4-methyl-1-piperazinyl)-2-oxoethyl]-N-[6-(4-pyridinyl)imidazo[1,2-a]pyridin-2-yl]benzamide |
| Purity: | ≥98% (HPLC) |
Potent and selective Dyrk1B kinase inhibitor
| Chemical Name: | 3-(2-Methyl-4-pyrimidinyl)-1-(phenylmethyl)-1H-pyrrolo[2,3-c]pyridine |
| Purity: | ≥98% (HPLC) |
Potent CK2A2 and CK2A1 inhibitor; also inhibits DYRK2
| Chemical Name: | N-[5-[[3-Cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methylphenyl]propanamide |
| Purity: | ≥98% (HPLC) |
Potent LMTK3 inhibitor
| Chemical Name: | 6-(Pyridin-4-yl)-3-(3-(trifluoromethoxy)phenyl)imidazo[1,2-b]pyridazine |
| Purity: | ≥98% (HPLC) |
