TRPM Blockers: Small Molecules and Peptides
9 results for "TRPM Blockers Small Molecules and Peptides" in Products
9 results for "TRPM Blockers Small Molecules and Peptides" in Products
TRPM Blockers: Small Molecules and Peptides
NMDA potentiator; also GABAA inhibitor and TRPM3 activator
| Chemical Name: | (3β)-3-(Sulfooxy)-pregn-5-en-20-one sodium salt |
Selective TRPM4 blocker
| Chemical Name: | 4-Chloro-2-[[2-(2-chlorophenoxy)acetyl]amino]benzoic acid |
| Purity: | ≥98% (HPLC) |
TRPM3 blocker
| Chemical Name: | 1-(2,4-Dihydroxyphenyl)-2-(4-methoxyphenyl)ethanone |
| Purity: | ≥98% (HPLC) |
TRPM8 blocker
| Chemical Name: | N-(4-Fluorophenyl)-3,4-dihydro-1-[4-(trifluoromethyl)phenyl]-2(1H)-isoquinolinecarboxamide |
| Purity: | ≥99% (HPLC) |
Potent and selective TRPM8 channel blocker
| Chemical Name: | N-(2-Aminoethyl)-N-[[3-methoxy-4-(phenylmethoxy)phenyl]methyl]-2-thiophenecarboxamide hydrochloride |
| Purity: | ≥99% (HPLC) |
TRPM8 blocker
| Chemical Name: | N-(3-Aminopropyl)-2-[(3-methylphenyl)methoxy]-N-(2-thienylmethyl)benzamide hydrochloride |
| Purity: | ≥99% (HPLC) |
Potent TRPM8 antagonist
| Chemical Name: | 3-[7-(Trifluoromethyl)-5-[2-(trifluoromethyl)phenyl]-1H-benzimidazol-2-yl]-1-oxa-2-azaspiro[4.5]dec-2-ene |
| Purity: | ≥98% (HPLC) |
Potent and selective TRPM8 antagonist; orally active
| Chemical Name: | 4-[[[3-Chloro-5-(trifluoromethyl)-2-pyridinyl][[4-(trifluoromethoxy)phenyl]methyl]amino]sulfonyl]benzoic acid |
| Purity: | ≥98% (HPLC) |
Potent and selective TRPM8 antagonist; active in vivo
| Chemical Name: | 6-[[[(S)-(3-Fluoro-2-pyridinyl)[3-fluoro-4-(trifluoromethoxy)phenyl]methyl]amino]carbonyl]-3-pyridinecarboxylic acid |
| Purity: | ≥98% (HPLC) |
