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Vanilloid R1/TRPV1: Small Molecules and Peptides

Vanilloid Receptor 1 (VR1) also known as TRPV1 (Transient Receptor Potential Vanilloid 1) and capsaicin receptor, is a 115 kDa integral membrane ion channel that has six transmembrane domains and contains intracellular N-and C-termini. Vanilloid Receptor 1 contributes to normal pain and temperature sensation and also has a sensory-effector function. By alternative splicing, at least three VR1 isoforms are known. The sequence of residues 4 - 21 of rat VR1 is 78% and 28% identical to that of mouse and human VR1, respectively.

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15 results for "Vanilloid R1/TRPV1 Small Molecules and Peptides" in Products

15 results for "Vanilloid R1/TRPV1 Small Molecules and Peptides" in Products

Vanilloid R1/TRPV1: Small Molecules and Peptides

Vanilloid Receptor 1 (VR1) also known as TRPV1 (Transient Receptor Potential Vanilloid 1) and capsaicin receptor, is a 115 kDa integral membrane ion channel that has six transmembrane domains and contains intracellular N-and C-termini. Vanilloid Receptor 1 contributes to normal pain and temperature sensation and also has a sensory-effector function. By alternative splicing, at least three VR1 isoforms are known. The sequence of residues 4 - 21 of rat VR1 is 78% and 28% identical to that of mouse and human VR1, respectively.

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Applications: WB

TRPV agonist

TRPV1 antagonist

Potent and selective TRPV1 competitive antagonist

Endogenous and non-selective CB agonist

Potent TRPV1 antagonist

Chloride channel blocker; TRPV1 modulator; RAD51 recombinase inhibitor

TRPV antagonist; also activator of ENaCδ

Reversible, competitive and potent TRPV1 antagonist

Potent and selective TRPV1 competitive antagonist

Potent and selective TRPV1 antagonist

Potent and selective TRPV1 antagonist

Potent TRPV1 antagonist

Potent and selective endogenous TRPV1 agonist

Potent TRPV agonist

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