Cannabinoid R1/CB1 Receptor Ligand Products
Cannabinoid Receptors are seven-pass transmembrane proteins that belong to the rhodopsin family of G protein-coupled receptors. There are at least two types of Cannabinoid receptors, CB1R and CB2R, which are activated by a family of endogenous arachidonic acid derivatives, such as the endocannabinoids and D9-THC. CB1R is expressed in the central nervous system and upper GI tract, while CB2R is expressed by selected neuronal cell types and hematopoietic cells.
2 results for "Cannabinoid R1/CB1 Receptor Ligand" in Products
2 results for "Cannabinoid R1/CB1 Receptor Ligand" in Products
Cannabinoid R1/CB1 Receptor Ligand Products
Cannabinoid Receptors are seven-pass transmembrane proteins that belong to the rhodopsin family of G protein-coupled receptors. There are at least two types of Cannabinoid receptors, CB1R and CB2R, which are activated by a family of endogenous arachidonic acid derivatives, such as the endocannabinoids and D9-THC. CB1R is expressed in the central nervous system and upper GI tract, while CB2R is expressed by selected neuronal cell types and hematopoietic cells.
Fluorescent cannabinoid ligand; fluorescent form of AM 251 (Cat. No. 1117)
| Chemical Name: | N-(Piperidin-1-yl)-5-(4-(4-(3-(5-carboxamidotetramethylrhodaminyl)propyl))phenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide |
| Purity: | ≥95% (HPLC) |
Potent and selective CB2 partial agonist; orally biovailable
| Chemical Name: | 3-Cyclopropyl-1-[[4-[6-[(1,1-dioxido-4-thiomorpholinyl)methyl]-5-fluoro-2-pyridinyl]phenyl]methyl]-2,4-imidazolidinedione hydrochloride |
| Purity: | ≥98% (HPLC) |
