Adenosine A3 Receptor Antagonists: Small Molecules and Peptides
Adenosine A3 Receptor (ADORA3) belongs to the family of adenosine receptors, which are G protein-coupled receptors involved in a variety of intracellular signaling pathways and physiological functions. ADORA3 mediates a sustained cardioprotective function during cardiac ischemia. It is involved in the inhibition of neutrophil degranulation in neutrophil-mediated tissue injury. ADORA3 has been implicated in both neuroprotective and neurodegenerative effects, and it may also mediate both cell proliferation and cell death.
4 results for "Adenosine A3 Receptor Antagonists Small Molecules and Peptides" in Products
4 results for "Adenosine A3 Receptor Antagonists Small Molecules and Peptides" in Products
Adenosine A3 Receptor Antagonists: Small Molecules and Peptides
Adenosine A3 Receptor (ADORA3) belongs to the family of adenosine receptors, which are G protein-coupled receptors involved in a variety of intracellular signaling pathways and physiological functions. ADORA3 mediates a sustained cardioprotective function during cardiac ischemia. It is involved in the inhibition of neutrophil degranulation in neutrophil-mediated tissue injury. ADORA3 has been implicated in both neuroprotective and neurodegenerative effects, and it may also mediate both cell proliferation and cell death.
Potent and selective A3 adenosine receptor antagonist
| Chemical Name: | N-[4-(3,5-Dimethylphenyl)-5-(4-pyridinyl)-2-thiazolyl]-3-pyridinecarboxamide dihydrochloride |
| Purity: | ≥98% |
Potent, highly selective hA3 receptor antagonist/inverse agonist
| Chemical Name: | (8R)-8-Ethyl-1,4,7,8-tetrahydro-4-methyl-2-(2,3,5-trichlorophenyl)-5H-imidazo[2,1-i]purin-5-one monohydrochloride |
| Purity: | ≥98% |
Highly potent and selective hA3 antagonist
| Chemical Name: | N-[9-Chloro-2-(2-furanyl)[1,2,4]-triazolo[1,5-c]quinazolin-5-yl]benzene acetamide |
| Purity: | ≥98% (HPLC) |
Potent, highly selective hA3 antagonist
| Chemical Name: | 1,4-Dihydro-2-methyl-6-phenyl-4-(phenylethynyl)-3,5-pyridinedicarboxylic acid 3-ethyl-5-[(3-nitrophenyl)methyl] ester |
| Purity: | ≥98% (HPLC) |
