GABA-A Receptor Modulators: Small Molecules and Peptides
Members of Cys-loop family of ligand-gated ion channels, the GABAA receptors are permeable to Cl-.
11 results for "GABA-A Receptor Modulators Small Molecules and Peptides" in Products
11 results for "GABA-A Receptor Modulators Small Molecules and Peptides" in Products
GABA-A Receptor Modulators: Small Molecules and Peptides
Members of Cys-loop family of ligand-gated ion channels, the GABAA receptors are permeable to Cl-.
Positive allosteric modulator of GABAA receptors
| Alternate Names: | 3a,5a-THPROG |
| Chemical Name: | (3α,5α)-3-Hydroxy-pregnan-20-one |
GABA-mimetic; selectively interacts with β2- and β3-subunit containing GABAA receptors
| Chemical Name: | (R)-1-(1-Phenylethyl)-1H-imidazole-5-carboxylic acid ethyl ester |
| Purity: | ≥98% (HPLC) |
Positive modulator of GABAA receptors; endogenous neurosteroid
| Chemical Name: | (3α,5α)-3,21-Dihydroxypregnan-20-one |
| Purity: | ≥95% (HPLC) |
Postitive allosteric modulator of GABAA receptors
| Chemical Name: | (3α,5β)-3-Hydroxy-pregnan-20-one |
Positive allosteric modulator of GABAA receptors; displays subunit selectivity
| Chemical Name: | 4-Chloro-N-[2-(2-thienyl)imidazo[1,2-a]pyridin-3-yl]benzamide |
| Purity: | ≥97% (HPLC) |
Potent positive allosteric modulator of GABAA receptors
| Alternate Names: | CCD 1042 |
| Chemical Name: | (3α,5α)-3-Hydroxy-3-methyl-pregnan-20-one |
GluK1 antagonist; inhibits carbonic anhydrase (CA) II and IV; also positive allosteric modulator of GABAA receptors
| Alternate Names: | Topamax |
| Chemical Name: | 2,3:4,5-Bis-O-(1-methylethylidene)-β-D-fructopyranose sulfamate |
| Purity: | ≥99% (HPLC) |
Allosteric modulator of GABAA receptors
| Alternate Names: | ICI 136753 |
| Chemical Name: | 4-(Butylamino)-1-ethyl-6-methyl 1H-pyrazolo[3,4b]pyridine-5-ethylcarboxylate hydrochloride |
| Purity: | ≥99% (HPLC) |
Ligand of the translocator protein (TSPO); also GABAA receptor potentiator
| Chemical Name: | 6-Chloro-2-N-ethyl-4-methyl-4-phenyl-4H-3,1-benzoxazin-2-amine hydrochloride |
| Purity: | ≥98% (HPLC) |
Subtype-selective GABAA modulator
| Chemical Name: | (Z)-1-[2-Chloro-2-(2,4-dichlorophenyl)ethenyl]-1H-1,2,4-triazole hydrochloride |
| Purity: | ≥99% (HPLC) |
KV7 channel activator; also GABAA modulator and indirect NMDA antagonist
| Alternate Names: | D 9998 |
| Chemical Name: | N-[2-Amino-6-[[4-fluorophenyl)methyl]amino]-3-pyridinyl]carbamic acid ethyl ester maleate |
| Purity: | ≥98% (HPLC) |
