Histamine H2 Receptor Antagonists: Small Molecules and Peptides
Histamine is a ubiquitous messenger molecule released from mast cells, enterochromaffin-like cells, and neurons. Its various actions are mediated by histamine receptors H1, H2, H3 and H4. HRH2 belongs to the family 1 of G protein-coupled receptors. Histamine H2 R is an integral membrane protein and stimulates gastric acid secretion. It also regulates gastrointestinal motility and intestinal secretion and is thought to be involved in regulating cell growth and differentiation. Alternatively spliced transcript variants encoding different isoforms have been found for this gene.
3 results for "Histamine H2 Receptor Antagonists Small Molecules and Peptides" in Products
3 results for "Histamine H2 Receptor Antagonists Small Molecules and Peptides" in Products
Histamine H2 Receptor Antagonists: Small Molecules and Peptides
Histamine is a ubiquitous messenger molecule released from mast cells, enterochromaffin-like cells, and neurons. Its various actions are mediated by histamine receptors H1, H2, H3 and H4. HRH2 belongs to the family 1 of G protein-coupled receptors. Histamine H2 R is an integral membrane protein and stimulates gastric acid secretion. It also regulates gastrointestinal motility and intestinal secretion and is thought to be involved in regulating cell growth and differentiation. Alternatively spliced transcript variants encoding different isoforms have been found for this gene.
Potent and selective H2 antagonist
| Purity: | ≥98% |
Potent, centrally active H2 antagonist
| Chemical Name: | N-[3-[3-(1-Piperidinylmethyl)phenoxy]propyl]-2-benzothiazolamine dimaleate |
H2 antagonist, I1 agonist
| Chemical Name: | N-Cyano-N'-methyl-N''-[2-[(5-methyl-1H-imidazol-4-yl)methyl]thio]ethyl]guanidine |
| Purity: | ≥99% (HPLC) |
