Histamine H3 Receptor Agonists: Small Molecules and Peptides
Histamine is a ubiquitous messenger molecule released from mast cells, enterochromaffin-like cells, and neurons. Its various actions are mediated by histamine receptors Histamine H1 R, Histamine H2 R, Histamine H3 R and Histamine H4 R. HRH3 encodes one of the histamine receptors (H3) which belongs to the family 1 of G protein-coupled receptors. Histamine H3 R is an integral membrane protein and can regulate neurotransmitter release. It can also increase voltage-dependent calcium current in smooth muscles and innervates the blood vessels and the heart in cardiovascular system.
4 results for "Histamine H3 Receptor Agonists Small Molecules and Peptides" in Products
4 results for "Histamine H3 Receptor Agonists Small Molecules and Peptides" in Products
Histamine H3 Receptor Agonists: Small Molecules and Peptides
Histamine is a ubiquitous messenger molecule released from mast cells, enterochromaffin-like cells, and neurons. Its various actions are mediated by histamine receptors Histamine H1 R, Histamine H2 R, Histamine H3 R and Histamine H4 R. HRH3 encodes one of the histamine receptors (H3) which belongs to the family 1 of G protein-coupled receptors. Histamine H3 R is an integral membrane protein and can regulate neurotransmitter release. It can also increase voltage-dependent calcium current in smooth muscles and innervates the blood vessels and the heart in cardiovascular system.
Endogenous histamine receptor agonist
| Chemical Name: | 2-(4-Imidazolyl)ethylamine dihydrochloride |
Potent, standard H3 agonist
| Chemical Name: | (R)-(-)-α-Methyl-1H-imidazole-4-ethanamine dihydrobromide |
| Purity: | ≥98% (HPLC) |
Standard H3 agonist. Also H4 agonist
| Chemical Name: | 4-(1H-Imidazol-4-ylmethyl)piperidine dihydrobromide |
Standard H3 and H4 agonist (H3 > H4)
| Chemical Name: | 5-[2-(Imidazol-4-yl)ethyl]isothiourea dihydrobromide |
| Purity: | ≥98% (HPLC) |
