Retinoic Acid Receptor Antagonists: Small Molecules and Peptides
Retinoic acid receptors (RARs) are nuclear hormone receptors of the NR1B class. The three subtypes of RARs include RARα, RARβ and RARγ.
8 results for "Retinoic Acid Receptor Antagonists Small Molecules and Peptides" in Products
8 results for "Retinoic Acid Receptor Antagonists Small Molecules and Peptides" in Products
Retinoic Acid Receptor Antagonists: Small Molecules and Peptides
Retinoic acid receptors (RARs) are nuclear hormone receptors of the NR1B class. The three subtypes of RARs include RARα, RARβ and RARγ.
High affinity pan-RAR antagonist
| Chemical Name: | 4-[2-[5,6-Dihydro-5,5-dimethyl-8-(4-methylphenyl)-2-naphthalenyl]ethynyl]benzoic acid |
| Purity: | ≥98% (HPLC) |
Selective RARα antagonist
| Chemical Name: | 4-[5-[8-(1-Methylethyl)-4-phenyl-2-quinolinyl]-1H-pyrrolo-2-benzoic acid |
| Purity: | ≥99% (HPLC) |
Selective RARβ antagonist
| Chemical Name: | 4-(7,8,9,10-Tetrahydro-5,7,7,10,10-pentamethyl-5H-benzo[e]naphtho[2,3-b][1,4]diazepin-13-yl)benzoic acid |
| Purity: | ≥97% (HPLC) |
Selective RARα antagonist
| Alternate Names: | BMS614 |
| Chemical Name: | 4-[[[5,6-Dihydro-5,5-dimethyl-8-(3-quinolinyl)-2-naphthalenyl]carbonyl]amino]benzoic acid |
| Purity: | ≥98% (HPLC) |
AGN 193109 synthesized to Ancillary Material Grade
| Chemical Name: | 4-[2-[5,6-Dihydro-5,5-dimethyl-8-(4-methylphenyl)-2-naphthalenyl]ethynyl]benzoic acid |
| Purity: | ≥98% |
High affinity and selective RARγ antagonist
| Chemical Name: | 4-[5-[3,5-Bis(1,1-dimethylethyl)phenyl]-1-[4-[(4-methyl-1-piperazinyl)carbonyl]phenyl]-1H-pyrazol-3-yl]benzoic acid |
| Purity: | ≥98% (HPLC) |
RARγ-selective antagonist
| Chemical Name: | 6-[2-(5,6,7,8-Tetrahydro-5,5,8,8-tetramethyl-2-naphthalenyl)-1,3-dithiolan-2-yl]-2-naphthalenecarboxylic acid |
| Purity: | ≥98% (HPLC) |
Selective RARβ/γ antagonist
| Chemical Name: | 4-[6-[(2-Methoxyethoxy)methoxy]-7-tricyclo[3.3.1.13,7]dec-1-yl-2-naphthalenyl)benzoic acid |
| Purity: | ≥98% (HPLC) |
