Vasopressin Receptor Antagonists: Small Molecules and Peptides
6 results for "Vasopressin Receptor Antagonists Small Molecules and Peptides" in Products
6 results for "Vasopressin Receptor Antagonists Small Molecules and Peptides" in Products
Vasopressin Receptor Antagonists: Small Molecules and Peptides
Selective vasopressin V1A antagonist
| Purity: | ≥95% (HPLC) |
Selective, orally active vasopressin V1A receptor antagonist
| Alternate Names: | Relcovaptan |
| Chemical Name: | (2S)-1-[[(2R,3S)-5-Chloro-3-(2-chlorophenyl)-1-[(3,4-dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-hydroxy-1H-indol-2-yl]carbonyl]-2-pyrrolidinecarboxamide |
| Purity: | ≥99% (HPLC) |
Potent and selective vasopressin V2 receptor antagonist; renoprotective and orally active
| Alternate Names: | OPC-41061 |
| Chemical Name: | N-[4-[(7-Chloro-2,3,4,5-tetrahydro-5-hydroxy-1H-1-benzazepin-1-yl)carbonyl]-3-methylphenyl]-2-methylbenzamide |
| Purity: | ≥98% (HPLC) |
Potent and selective V1B receptor antagonist; orally bioavailable
| Chemical Name: | 2-(3-Chloro-4-fluorophenyl)-N-(1-methylethyl)-6-[3-(4-morpholinyl)propoxy]-4-oxo-pyrido[2,3-d]pyrimidine-3(4H)-acetamide hydrochloride |
| Purity: | ≥98% (HPLC) |
Very high affinity vasopressin V1A and V2 antagonist; orally bioavailable
| Chemical Name: | N-[4-[(4,5-Dihydro-2-methylimidazo[4,5-d][benzazepin-6(1H)-yl)carbonyl]phenyl-[1,1'-biphenyl]-2-carboxamide hydrochloride |
| Purity: | ≥98% (HPLC) |
Potent and selective vasopressin V1B antagonist
| Alternate Names: | Nelivaptan |
| Chemical Name: | (2S,4R)-1-[(3R)-5-Chloro-1-[(2,4-dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-(2-methoxyphenyl)-2-oxo-1H-indol-3-yl]-4-hydroxy-N,N-dimethyl-2-pyrrolidinecarboxamide |
| Purity: | ≥98% (HPLC) |
