GABA-B Receptor Antagonists: Small Molecules and Peptides
GABAB receptors are metabotropic G-protein-coupled receptors (GPCRs). They are responsible for mediating the inhibitory effects of GABA and ionotropic GABAA and GABAA-ρ receptors.
9 results for "GABA-B Receptor Antagonists Small Molecules and Peptides" in Products
9 results for "GABA-B Receptor Antagonists Small Molecules and Peptides" in Products
GABA-B Receptor Antagonists: Small Molecules and Peptides
GABAB receptors are metabotropic G-protein-coupled receptors (GPCRs). They are responsible for mediating the inhibitory effects of GABA and ionotropic GABAA and GABAA-ρ receptors.
Potent and selective GABAB antagonist
| Chemical Name: | (2S)-3-[[(1S)-1-(3,4-Dichlorophenyl)ethyl]amino-2-hydroxypropyl](phenylmethyl)phosphinic acid hydrochloride |
| Purity: | ≥98% (HPLC) |
Selective GABAB antagonist
| Chemical Name: | (RS)-3-Amino-2-(4-chlorophenyl)propylsulfonic acid |
| Purity: | ≥99% |
GABAB antagonist; displays activity at presynaptic receptors
| Chemical Name: | (3-Aminopropyl)ethylphosphinic acid hydrochloride |
| Purity: | ≥99% (HPLC) |
Potent and selective GABAB antagonist
| Chemical Name: | [S-(R*,R*)]-[3-[[1-(3,4-Dichlorophenyl)ethyl]amino]-2-hydroxypropyl](cyclohexylmethyl) phosphinic acid |
| Purity: | ≥96% (HPLC) |
Selective GABAB antagonist; more potent than Saclofen (Cat. No. 0246)
| Chemical Name: | (RS)-3-Amino-2-(4-chlorophenyl)-2-hydroxypropyl-sulfonic acid |
Selective GABAB antagonist; brain penetrant
| Chemical Name: | (3-Aminopropyl)(cyclohexylmethyl)phosphinic acid |
Selective GABAB antagonist; brain penetrant
| Chemical Name: | (3-Aminopropyl)(diethoxymethyl)phosphinic acid |
Potent and selective GABAB antagonist
| Chemical Name: | 3-[[(3,4-Dichlorophenyl)methyl]amino]propyl] diethoxymethyl)phosphinic acid |
| Purity: | ≥98% (HPLC) |
Selective and competitive GABAB antagonist; orally bioavailable
| Chemical Name: | (2S)-(+)-5,5-Dimethyl-2-morpholineacetic acid |
| Purity: | ≥98% |
