Prostanoid Receptor Antagonists: Small Molecules and Peptides
13 results for "Prostanoid Receptor Antagonists Small Molecules and Peptides" in Products
13 results for "Prostanoid Receptor Antagonists Small Molecules and Peptides" in Products
Prostanoid Receptor Antagonists: Small Molecules and Peptides
Selective EP1 receptor antagonist
Chemical Name: | 8-Chloro-dibenzo(Z)[b,f][1,4]oxazepine-10(11H)-carboxylic acid, 2-acetylhydrazide |
Purity: | ≥99% (HPLC) |
Dual TP/DP2 (CRTH2) receptor antagonist
Alternate Names: | Ramatroban |
Chemical Name: | (3R)-3-[[(4-Fluorophenyl)sulfonyl]amino]-1,2,3,4-tetrahydro-9H-carbazole-9-propanoic acid |
Purity: | ≥99% (HPLC) |
EP1 receptor antagonist
Chemical Name: | 4-[[[2,3-Dihydro-6-[(2-methylpropyl)[(4-methyl-2-thiazolyl)sulfonyl]amino]-1H-indene-5yl]oxy]methyl]benzoic acid |
Purity: | ≥98% (HPLC) |
Potent and selective EP2 receptor antagonist
Chemical Name: | 1-(4-Fluorobenzoyl)-3-[[(6-methoxy-2-naphthalenyl)oxy]methyl]-3-azetidinecarboxylic acid |
Purity: | ≥98% (HPLC) |
Selective EP4 receptor antagonist
Chemical Name: | N-[[4'-[[3-Butyl-1,5-dihydro-5-oxo-1-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-4-yl]methyl][1,1'-biphenyl]-2-yl]sulfonyl]-3-methyl-2-thiophenecarboxamide |
Purity: | ≥99% (HPLC) |
Potent EP1 receptor antagonist
Chemical Name: | 8-Chloro-2-[3-[(2-furanylmethyl)thio]-1-oxopropyl]-dibenz(Z)[b,f][1,4]oxazepine-10(11H)-carboxylic acid hydrazide |
Purity: | ≥98% (HPLC) |
Potent dual CRTH2 and prostaglandin D2 (PGD2) receptor antagonist
Chemical Name: | 5-Chloro-4-[2-[[(2-chloro-4-cyclopropylphenyl)sulfonyl]amino]-4-[[(1,1-dimethylethyl)amino]carbonyl]phenoxy]-2-fluorobenzeneacetic acid |
Purity: | ≥98% (HPLC) |
Potent and selective prostaglandin D2 receptor antagonist
Chemical Name: | (3R)-4-[(4-Chlorophenyl)methyl]-7-fluoro-1,2,3,4-tetrahydro-5-(methylsulfonyl)cyclopent[b]indole-3-acetic acid |
Purity: | ≥98% (HPLC) |
Potent and highly selective EP3 antagonist
Chemical Name: | N-[(5-Bromo-2-methoxyphenyl)sulfonyl]-3-[2-(2-naphthalenylmethyl)phenyl]-2-propenamide |
Purity: | ≥99% (HPLC) |
High affinity and selective EP4 antagonist
Alternate Names: | PGN 1531 |
Chemical Name: | 4-[[4-(5-Methoxy-2-pyridinyl)phenoxy]methyl]-5-methyl-N-[(2-methylphenyl)sulfonyl]-2-furancarboxamide hydrochloride |
Purity: | ≥98% (HPLC) |
Potent thromboxane A2 (TP) antagonist
Alternate Names: | terutroban |
Chemical Name: | (6R)-6-[[(4-Chlorophenyl)sulfonyl]amino]-5,6,7,8-tetrahydro-2-methyl-1-naphthalenepropanoic acid |
Purity: | ≥98% (HPLC) |
High affinity and selective EP4 antagonist
Chemical Name: | 4-Cyano-2-[[2-(4-fluoro-1-naphthalenyl)-1-oxopropyl]amino]benzenebutanoic acid |
Purity: | ≥98% (HPLC) |
Potent and selective EP3 antagonist; antiplatelet and antithrombotic
Chemical Name: | (2E)-3-[1-[(2,4-Dichlorophenyl)methyl]-5-fluoro-3-methyl-1H-indol-7-yl]-N-[(4,5-dichloro-2-thienyl)sulfonyl]-2-propenamide |
Purity: | ≥98% (HPLC) |