TRPV Antagonists: Small Molecules and Peptides
17 results for "TRPV Antagonists Small Molecules and Peptides" in Products
17 results for "TRPV Antagonists Small Molecules and Peptides" in Products
TRPV Antagonists: Small Molecules and Peptides
TRPV antagonist; also activator of ENaCδ
| Chemical Name: | N-[2-(4-Chlorophenyl)ethyl]-1,3,4,5-tetrahydro-7,8-dihydroxy-2H-2-benzazepine-2-carbothioamide |
| Purity: | ≥99% (HPLC) |
Potent and selective TRPV4 antagonist; orally active
| Chemical Name: | 3-([1,4'-Bipiperidin]-1'-ylmethyl)-7-bromo-N-(1-phenylcyclopropyl)-2-[3-(trifluoromethyl)phenyl]-4-quinolinecarboxamide |
| Purity: | ≥98% (HPLC) |
Potent and selective TRPV1 competitive antagonist
| Chemical Name: | (2E)-N-(2,3-Dihydro-1,4-benzodioxin-6-yl)-3-[4-(1,1-dimethylethyl)phenyl]-2-propenamide |
| Purity: | ≥98% (HPLC) |
Potent TRPV1 antagonist
| Chemical Name: | N-[4-[[6-[4-(Trifluoromethyl)phenyl]-4-pyrimidinyl]oxy]-2-benzothiazolyl]acetamide |
| Purity: | ≥98% (HPLC) |
Potent and selective TRPV4 antagonist
| Chemical Name: | 2-Methyl-1-[3-(4-morpholinyl)propyl]-5-phenyl-N-[3-(trifluoromethyl)phenyl]-1H-pyrrole-3-carboxamide |
| Purity: | ≥99% (HPLC) |
Potent and selective TRPV1 competitive antagonist
| Chemical Name: | 4'-Chloro-3-methoxycinnamanilide |
| Purity: | ≥99% (HPLC) |
Selective TRPV3 antagonist; brain penetrant
| Chemical Name: | (αS)-α-[cis-3-Hydroxy-3-methyl-1-[4-(trifluoromethyl)-2-pyridinyl]cyclobutyl]-2-pyridinemethanol |
| Purity: | ≥98% (HPLC) |
Selective TRPV4 antagonist
| Chemical Name: | 2,4-Dichloro-N-isopropyl-N-(2-isopropylaminoethyl)benzenesulfonamide |
TRPV1 antagonist
| Chemical Name: | 4-(3-Chloro-2-pyridinyl)-N-[4-(1,1-dimethylethyl)phenyl]-1-piperazinecarboxamide |
| Purity: | ≥98% (HPLC) |
Potent and selective TRPV1 antagonist
| Chemical Name: | 3,6-Dihydro-3'-(trifluoromethyl)-N-[4-[(trifluoromethyl)sulfonyl]phenyl]-[1(2H),2'-bipyridine]-4-carboxamide |
| Purity: | ≥99% (HPLC) |
Selective TRPV2 antagonist
| Chemical Name: | N-(2-Furanylmethyl)-3-[[4-(methylpropylamino)-6-(trifluoromethyl)-2-pyrimidinyl]thio]propanamide |
| Purity: | ≥98% (HPLC) |
Potent and selective TRPV4 antagonist
| Chemical Name: | N-[4-[[4-(1-Methylethyl)-1-piperazinyl]sulfonyl]phenyl]-2-nitro-4-(trifluoromethyl)benzamide hydrochloride |
| Purity: | ≥99% (HPLC) |
Non-selective CaV2.1 and 2.2 blocker; also blocks TRPV channels
| Chemical Name: | Ammoniated ruthenium oxychloride |
Reversible, competitive and potent TRPV1 antagonist
| Chemical Name: | 4-[3-(Trifluoromethyl)-2-pyridinyl]-N-[5-(trifluoromethyl)-2-pyridinyl]-1-piperazinecarboxamide |
| Purity: | ≥99% (HPLC) |
Potent TRPV1 antagonist
| Chemical Name: | N-5-Isoquinolinyl-N'-[[(4-(trifluoromethyl)phenyl]methyl]urea |
| Purity: | ≥98% (HPLC) |
Potent and selective TRPV1 antagonist
| Chemical Name: | 3-Amino-5-[[2-[(2-methoxyethyl)amino]-6-[4-(trifluoromethyl)phenyl]-4-pyrimidinyl]oxy]-2(1H)-quinoxalinone |
| Purity: | ≥97% (HPLC) |
Antiallergic; inhibits inflammatory mediator release from mast cells
| Chemical Name: | 2-[[3-(3,4-Dimethoxyphenyl)-1-oxo-2-propenyl]amino]benzoic acid |
| Purity: | ≥99% (HPLC) |
