Group I mGluR Antagonists: Small Molecules and Peptides
17 results for "Group I mGluR Antagonists Small Molecules and Peptides" in Products
17 results for "Group I mGluR Antagonists Small Molecules and Peptides" in Products
Group I mGluR Antagonists: Small Molecules and Peptides
Competitive group I mGlu antagonist; also weak group II agonist
Alternate Names: | (S)-4CPG |
Purity: | ≥99% (HPLC) |
Potent and selective group I mGlu antagonist
Alternate Names: | UPF 523 |
Chemical Name: | (RS)-1-Aminoindan-1,5-dicarboxylic acid |
Purity: | ≥98% (HPLC) |
Potent group I mGlu antagonist
Chemical Name: | N-Phenyl-7-(hydroxyimino)cyclopropa[b]chromen-1a-carboxamide |
Purity: | ≥98% (HPLC) |
Group I mGlu antagonist
Chemical Name: | N-tricyclo[3.3.1.13,7]dec-1-yl-2-quinoxalinecarboxamide |
Purity: | ≥99% (HPLC) |
Potent mGlu5 antagonist; also positive allosteric modulator of mGlu4 receptors
Chemical Name: | 2-Methyl-6-(phenylethynyl)pyridine hydrochloride |
Purity: | ≥99% (HPLC) |
Selective non-competitive mGlu1 antagonist
Chemical Name: | 7-(Hydroxyimino)cyclopropa[b]chromen-1a-carboxylate ethyl ester |
Purity: | ≥99% (HPLC) |
Highly potent, mGlu1-selective non-competitive antagonist
Chemical Name: | (3,4-Dihydro-2H-pyrano[2,3-b]quinolin-7-yl)-(cis-4-methoxycyclohexyl)-methanone |
Purity: | ≥98% |
Selective mGlu1a antagonist
Chemical Name: | (S)-(+)-α-Amino-4-carboxy-2-methylbenzeneacetic acid |
Purity: | ≥99% (HPLC) |
Non-selective mGlu antagonist; disodium salt of (RS)-MCPG (Cat. No. 0336)
Chemical Name: | (RS)-α-Methyl-4-carboxyphenylglycine disodium salt |
Purity: | ≥99% (HPLC) |
Non-selective mGlu antagonist; active isomer of (RS)-MCPG (Cat. No. 0336)
Chemical Name: | (S)-α-Methyl-4-carboxyphenylglycine |
Purity: | ≥99% (HPLC) |
Selective mGlu1 antagonist
Chemical Name: | 6-Methoxy-N-(4-methoxyphenyl)-4-quinazolinamine hydrochloride |
Purity: | ≥99% |
mGlu1 inverse agonist
Chemical Name: | (3aS,6aS)-Hexahydro-5-methylene-6a-(2-naphthalenylmethyl)-1H-cyclopenta[c]furan-1-one |
Purity: | ≥98% |
Potent and selective mGlu5 antagonist
Chemical Name: | 3-((2-Methyl-1,3-thiazol-4-yl)ethynyl)pyridine hydrochloride |
Purity: | ≥99% (HPLC) |
Non-selective mGlu antagonist
Chemical Name: | (RS)-α-Methyl-4-carboxyphenylglycine |
Purity: | ≥99% (HPLC) |
High affinity human mGlu5 antagonist
Chemical Name: | 3-[2-(6-Methyl-2-pyridinyl)ethynyl]-2-cyclohexene-1-one O-methyloxime |
Purity: | ≥98% |
Potent and selective mGlu5 antagonist; brain penetrant
Chemical Name: | 3-Fluoro-5-[3-(5-fluoro-2-pyridinyl)-1,2,4-oxadiazol-5-yl]benzonitrile |
Purity: | ≥98% (HPLC) |
mGlu5 antagonist; orally bioavailable and brain penetrant
Chemical Name: | 4-[5-[(1R)-1-[5-(3-Chlorophenyl)-3-isoxazolyl]ethoxy]-4-methyl-4H-1,2,4-triazol-3-yl]pyridine |
Purity: | ≥98% (HPLC) |