Multidrug Transporter Inhibitors Products
12 results for "Multidrug Transporter Inhibitors" in Products
12 results for "Multidrug Transporter Inhibitors" in Products
Multidrug Transporter Inhibitors Products
Potent inhibitor of multidrug and toxin extrusion (MATE) transporters; also DHFR and STAT3 inhibitor
| Chemical Name: | 5-(4-Chlorophenyl)-6-ethyl-2,4-pyrimidinediamine |
| Purity: | ≥99% |
Potent and selective BCRP inhibitor
| Chemical Name: | (3S,6S,12aS)-1,2,3,4,6,7,12,12a-Octahydro-9-methoxy-6-(2-methylpropyl)-1,4-dioxopyrazino[1',2':1,6]pyrido[3,4-b]indole-3-propanoic acid 1,1-dimethylethyl ester |
| Purity: | ≥99% (HPLC) |
MRP and OAT3 inhibitor
| Chemical Name: | 4-(Dipropylsulfamoyl)benzoic acid |
| Purity: | ≥98% (HPLC) |
P-gp and BCRP inhibitor
| Alternate Names: | GF 120918 |
| Chemical Name: | N-[4-[2-(3,4-Dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)ethyl]phenyl]-9,10-dihydro-5-methoxy-9-oxo-4-acridinecarboxamide hydrochloride |
| Purity: | ≥98% (HPLC) |
Inhibitor of P-gp-mediated MDR
| Chemical Name: | 6-[(2S,4R,6E)-4-methyl-2-(methylamino)-3-oxo-6-octenoic acid]-7-L-valine-cyclosporin A |
| Purity: | ≥98% |
P-gp inhibitor
| Chemical Name: | 4-(3,4-Dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)-N-2[2-(3,4-dimethoxyphenyl)ethyl]-6,7-dimethoxy-2-quinazolinamine hydrochloride |
| Purity: | ≥98% (HPLC) |
High affinity P-gp inhibitor
| Alternate Names: | LY 335979 |
| Chemical Name: | (αR)-4-[(1aα,6α,10bα)-1,1-Difluoro-1,1a,6,10b-tetrahydrodibenzo[a,e]cyclopropa[c]cyclohepten-6-yl]-α-[(5-quinolinyloxy)methyl]-1-piperazineethanol trihydrochloride |
| Purity: | ≥97% (HPLC) |
Selective BCRP inhibitor
| Chemical Name: | N-[4-(2-Hydroxyethyl)phenyl]-2-[(4-nitrobenzoyl)amino]benzamide |
| Purity: | ≥98% (HPLC) |
Potent P-glycoprotein (P-gp) inhibitor
| Chemical Name: | N-[2-[[[4-[2-(3,4-dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)ethyl]phenyl]amino]carbonyl]-4,5-dimethoxyphenyl]-3-quinolinecarbxamide dihydrochloride |
| Purity: | ≥98% (HPLC) |
Selective MRP4 inhibitor
| Chemical Name: | 5-[(2-Benzothiazolylthio)methyl]-2,4-dihydro-4-methyl-3H-1,2,4-triazole-3-thione |
| Purity: | ≥98% |
Potent CysLT1 (LTD4) inverse agonist. Also MRP1 inhibitor
| Alternate Names: | L-660711 |
| Chemical Name: | 3-[[[3-[(1E)-2-(7-Chloro-2-quinolinyl)ethenyl]phenyl][[3-(dimethylamino)-3-oxopropyl]thio]methyl]thio]propanoic acid |
Selective MRP1 and P-gp inhibitor
| Chemical Name: | N-[3-(4-Morpholinyl)propyl]-5,7-diphenylpyrazolo[1,5-a]pyrimidine-3-carboxamide |
| Purity: | ≥95% |
